Cell-permeable. A dipeptide that acts as a selective and reversible PPARγ antagonist (KD ~ 8 μM). Shown to inhibit the agonist activity of Rosiglitazone (100 nM) in a dose-dependent manner (IC50= 31.9 μM) in transfected COS-7 cells.
| A.G. Scientific, Inc. | |
|---|---|
| Product Category | Biological Materials |
| Product Number | P-2406 |
| Product Name | PPARγ Antagonist, G3335 |