Lapatinib is a potent inhibitor of EGFR kinase (Ki = 3 nM), ErbB-2 kinase (Ki = 13 nM), ErbB-4 kinase (Ki = 347 nM). Lapatinib can restore tamoxifen sensitivity in tamoxifen-resistant,
| A.G. Scientific, Inc. | |
|---|---|
| Product Category | Biological Materials |
| Product Number | L-2371 |
| Product Name | Lapatinib Ditosylate (Tykerb, Tyverb, GW-572016) |