A.G. Scientific, Inc. Lapatinib Ditosylate (Tykerb, Tyverb, GW-572016) L-2371

Description
Lapatinib is a potent inhibitor of EGFR kinase (Ki = 3 nM), ErbB-2 kinase (Ki = 13 nM), ErbB-4 kinase (Ki = 347 nM). Lapatinib can restore tamoxifen sensitivity in tamoxifen-resistant, ER-positive breast cancer models.
Description
Lapatinib is a potent inhibitor of EGFR kinase (Ki = 3 nM), ErbB-2 kinase (Ki = 13 nM), ErbB-4 kinase (Ki = 347 nM). Lapatinib can restore tamoxifen sensitivity in tamoxifen-resistant, ER-positive breast cancer models.

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San Diego, CA, USA
Lapatinib Ditosylate (Tykerb, Tyverb, GW-572016)
L-2371
Lapatinib Ditosylate (Tykerb, Tyverb, GW-572016) L-2371
Lapatinib is a potent inhibitor of EGFR kinase (Ki = 3 nM), ErbB-2 kinase (Ki = 13 nM), ErbB-4 kinase (Ki = 347 nM). Lapatinib can restore tamoxifen sensitivity in tamoxifen-resistant, ER-positive breast cancer models.

Lapatinib is a potent inhibitor of EGFR kinase (Ki = 3 nM), ErbB-2 kinase (Ki = 13 nM), ErbB-4 kinase (Ki = 347 nM). Lapatinib can restore tamoxifen sensitivity in tamoxifen-resistant, ER-positive breast cancer models.

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Technical Specifications

  A.G. Scientific, Inc.
Product Category Biological Materials
Product Number L-2371
Product Name Lapatinib Ditosylate (Tykerb, Tyverb, GW-572016)
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