A.G. Scientific, Inc. 1-Azakenpaullone A-1312

Description
Analog of kenpaullone acting as a potent and ATP-competitive inhibitor of GSK-3β (IC50=18 nM). Displays ~100-200 fold greater selectivity on GSK-3Beta than over CDK1/cyclin B and CDK5/p25 (IC50=2.0 μM and 4.2 μM, respectively).
Description
Analog of kenpaullone acting as a potent and ATP-competitive inhibitor of GSK-3β (IC50=18 nM). Displays ~100-200 fold greater selectivity on GSK-3Beta than over CDK1/cyclin B and CDK5/p25 (IC50=2.0 μM and 4.2 μM, respectively).

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Product
Description
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A.G. Scientific, Inc.
San Diego, CA, USA
1-Azakenpaullone
A-1312
1-Azakenpaullone A-1312
Analog of kenpaullone acting as a potent and ATP-competitive inhibitor of GSK-3β (IC50=18 nM). Displays ~100-200 fold greater selectivity on GSK-3Beta than over CDK1/cyclin B and CDK5/p25 (IC50=2.0 μM and 4.2 μM, respectively).

Analog of kenpaullone acting as a potent and ATP-competitive inhibitor of GSK-3β (IC50=18 nM). Displays ~100-200 fold greater selectivity on GSK-3Beta than over CDK1/cyclin B and CDK5/p25 (IC50=2.0 μM and 4.2 μM, respectively).

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Technical Specifications

  A.G. Scientific, Inc.
Product Category Biological Materials
Product Number A-1312
Product Name 1-Azakenpaullone
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